Azelnidipine

Name: Azelnidipine
Brand: Jinan Shenghe Chemical Co., Ltd.

CAS 123524-52-7C33H34N4O6MW 582.6

Azelnidipine (CAS No. 123524-52-7) is supplied by Jinan Shenghe Chemical Co., Ltd. with a typical purity of 按批次COA提供(不公开发布). Main applications include Pharmaceutical Intermediates & APIs. Bulk quantities are available with COA; purity and packaging are subject to batch COA and order confirmation.

Specifications

CAS Number123524-52-7

Molecular FormulaC33H34N4O6

Molecular Weight582.6

Melting Point193-195

LogP5.18

Purity按批次COA提供(不公开发布)

Packaging按订单/批次确认(不公开发布)

ApplicationsPharmaceutical Intermediates & APIs

CategoryPharmaceutical Intermediates & APIs

Where it is used

Pharmaceutical Intermediates & APIs

Packaging & Supply

Packaging按订单/批次确认(不公开发布)

Purity按批次COA提供(不公开发布)

StorageSealed, cool and dry place

Lead TimeIn stock / per order

Documents & Support

COA provided with every batch; MSDS and technical documents available on request. Email us with product name and CAS number for a quote within one business day.

Frequently Asked Questions

What is the CAS number of Azelnidipine?

The CAS number of Azelnidipine is 123524-52-7.

What purity and packaging are available?

Typical purity is 按批次COA提供(不公开发布), supplied in 按订单/批次确认(不公开发布), with COA provided.

What are the applications of Azelnidipine?

Main applications include Pharmaceutical Intermediates & APIs.

How do I buy Azelnidipine or get a quote?

Email info@591daili.com or reach us on WhatsApp with the product name, CAS number and required quantity; quotes within one business day. Supplier: Jinan Shenghe Chemical Co., Ltd..

PubChem Public Data

Description

Azelnidipine · CAS 123524-52-7 · C33H34N4O6. UNII PV23P19YUG. Melting Point: 193-195; LogP: 5.18.

Identification

CAS Registry Number	123524-52-7
PubChem CID	65948
Molecular formula	C33H34N4O6
IUPAC name	3-O-(1-benzhydrylazetidin-3-yl) 5-O-propan-2-yl 2-amino-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate
UNII (FDA)	PV23P19YUG

Computed Descriptors

Molecular Weight	582.6
XLogP3	6
Hydrogen Bond Donor Count	2
Hydrogen Bond Acceptor Count	9
Rotatable Bond Count	10
Exact Mass	582.24783482
Monoisotopic Mass	582.24783482
Topological Polar Surface Area	140
Heavy Atom Count	43
Formal Charge	0

Physical & Chemical Properties

Melting Point	193-195
LogP	5.18

Physical description & handling notes

Insoluble in water

GHS Hazard Classification

Reported hazard statements	H302 (100%), H318 (95.1%)

H302 (100%): Harmful if swallowed [Warning Acute toxicity, oral]

H318 (95.1%): Causes serious eye damage [Danger Serious eye damage/eye irritation]

Documented Uses

For the treatment of hypertension.
Oral ingestion of azelnidipine demonstrates rapid and dose-dependent absorption.
In one study, following a single 4mg oral dose of 14C-labeled azelnidipine in humans, about 26% of the drug was thought to br excreted in the urine and 63% in the feces during the 1 week period post administration.
In a Chinese study examining the pharmacokinetics of the drug, the volume of distribution was found to be 1749 +/- 964.
Azelnidipine is widely bound to human plasma proteins (90%–91%).
Like most members of its class, azelnidipine primarily undergoes first-pass hepatic metabolism. Azelnidipine is metabolized by hepatic cytochrome P450 (CYP) 3A4 and has no active metabolite product. It may interact with other drugs or compounds that are substrates for this enzyme. Azelnidipine is lipophilic and has a potent affinity for membranes of vascular smooth muscle cells.

Synonyms

Azelnidipine; 123524-52-7; Calblock; CS-905; DTXSID3020120; Azelnidipino; PV23P19YUG; CS905; DTXCID50120; azelnidipinum; RefChem:560476; Azelnidipine [INN]; CS 905; MFCD00865803; C33H34N4O6; HMS3651D18

Frequently Asked Questions

What are the CAS number and molecular formula of Azelnidipine?

CAS 123524-52-7; molecular formula C33H34N4O6; molecular weight — g/mol.

What other names is Azelnidipine known by?

Azelnidipine, 123524-52-7, Calblock, CS-905, DTXSID3020120, Azelnidipino.

Is Azelnidipine classified as hazardous?

Hazard statements reported: H302, H318.

What are the key physical properties of Azelnidipine?

Melting Point: 193-195; LogP: 5.18.

Facts on this page are taken from PubChem (US National Library of Medicine) and Wikidata. Grade-specific data — assay, moisture, particle size, packaging, shelf life — is issued per batch on the COA and is not published here.

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